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Synthesis of thienopyridine derivatives and its anti-platelet activity in vivo

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Author:
No author available
Journal Title:
ACTA PHARMACEUTICA SINICA
Issue:
1
DOI:
No doi available
Key Word:
噻吩并四氢吡啶衍生物;合成;ADP受体拮抗剂;抗血小板聚集

Abstract: 为了寻找新型的ADP受体拮抗剂类抗血栓药物,合成了18个未见文献报道的噻吩并四氢吡啶衍生物、化合物结构经1H NMR和MS确证.大鼠体内抗血小板聚集活性研究表明,化合物CI的活性优于阳性对照药噻氯匹定,值得进一步深入研究;化合物A4、B2、C4和C7均有不同程度的抑制血小板聚集的活性.

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